產(chǎn)品屬性：
產(chǎn)品名稱 | Raloxifene 6-Glucuronide |
規(guī)格 | 1mg |
貨號 | EY-01Y14557 |
Cas No.: 174264-50-7
別名: N/A
化學名: N/A
分子式: C34H35NO10S
分子量: 649.7
溶解度: Soluble in DMSO
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述：
Raloxifene 6-glucuronide is a metabolite of the selective estrogen receptor modulator raloxifene . It is formed from raloxifene via the UDP-glucuronosyltransferase (UGT) isoforms UGT1A1 and UGT1A8. It binds to the estrogen receptor with an IC50 value of 290 nM. Unlike raloxifene, raloxifene 6-glucuronide does not inhibit the voltage-gated potassium channel Kv4.3.
特別提醒公司產(chǎn)品僅供科研使用
